Introduction
INTRODUCTION
Programme
Programme
Registration
Registration
Attendee Information
Attendee Information
Venue
VENUE
Partners
Partners
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Wednesday, September 7, 2022
12:00 - 17:00 Arrivals & Registration
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14:30 - 14:45 Conference opening
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14:45 - 16:30
Block of Lectures I
Chairs: dr. ROSS JANSEN-VAN VUUREN; assoc. prof. OLDŘICH FARSA
14:45 - 15:15 JANSEN-VAN VUUREN, R. (University of Ljubljana, Slovenia): Sustainable Approaches to the Preparation of Isotope-labelled Pharmaceuticals
15:15 - 15:45 SARKER, S. (Liverpool John Moores University, UK): Antimicrobial activity of Ruta chalepensis: A resazurin assay and scanning electron microscopy-based approach
15:45 - 16:00 FARSA, O. (Masaryk University, Czech republic): Aromatic Schiff bases as aminopeptidase N inhibitors
16:00 - 16:15 BRÁZDOVÁ, M. (Masaryk University, Czech republic): G-quadruplexes recognition by p53 family and modulation by ligands -
16:15 Welcome drink
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Thursday, September 8, 2022
9:00 - 10:45
Block of Lectures II
Chairs: assoc. prof. MARC OLSEN; assoc. prof. FILS ANDRIAMAINTY
9:00 - 9:30 OLSEN, M. (Midwestern University, USA): Design and Synthesis of Aspartyl(asparaginyl)-beta-hydroxylases for Treatment of Cancer
9:30 - 10:00 MALÍK, I. (Comenius University Bratislava, Slovakia): Synthesis and In Vitro Antimicrobial Activity of Some Hybrid Compounds Containing a Phenylcarbamic Acid Structural Motif
10:00 - 10:30 ŠVESTKA, D. (Masaryk University, Czech republic): Perhaloacetaldehydes in the enantioselective organocatalyzed fridel-crafts alkylation: reaction conditions development
10:30 - 10:45 NÁDASKÁ, D. (Comenius University Bratislava, Slovakia): Preliminary Investigation of Structure–Activity Relationships for Several Groups of Janus Kinase Inhibitors Using a Chemometric Principal Component Analysis -
10:45 - 11:15 Coffee break
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11:15 - 12:30
Block of Lectures III
Chairs: dr. ZUZANA HOLUBCOVÁ; assoc. prof. IVAN MALÍK
11:15 - 11:45 HOLUBCOVÁ, Z. (Masaryk University, Czech republic): Translating embryological research into clinical practice in assisted reproduction - benefits and limits of pharmacological intervention
11:45 - 12:00 KUCHYNKA, M. (Masaryk University, Czech republic): Imaging of elements and proteins in biological tissues: medical and pharmaceutical applications
12:00 - 12:15 PELCOVÁ, M. (Masaryk University, Czech republic): Pharmacokinetic profiling via dried blood spot sampling method
12:15 - 12:30 HAVRÁNKOVÁ, E. (Masaryk University, Czech republic): Novel 1,3,5-triazinyl aminobenzenesulfonamides as potent anti-VRE agents -
12:30 - 13:45 Lunch Break (arranged individually)
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13:45-15:30
Block of Lectures IV
Chairs: prof. RUDI H. ETTRICH; prof. PETER MIKUŠ
13:45 - 14:30 ETTRICH, R. H. (Larkin University, USA): Computational modeling of 3’-phosphoadenosine 5’- phosphosulfate synthase PAPSS
14:30 - 15:00 ŠMEJKAL, K. (Masaryk University, Czech republic): Prenylated phenolics as pleiotropic bioactive substances
15:00 - 15:15 DULEBA, J. (Nicholas Copernicus University, Poland): The effect of the 'catalytic triangle' on the lipase activity
15:15 - 15:30 VYLETELOVÁ, V. (Comenius University Bratislava, Slovakia): The combined treatment of methotrexate with carnosic acid influences hepatic mRNA expression of inflammatory and antioxidant genes in model of adjuvant artritis in rat -
15:30 - 16:00 Coffee break
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16:00 - 18:30
Block of lectures V
Chairs: assoc. prof. RADKA OPATŘILOVÁ; dr. PETR CHYTIL
16:00 - 16:45 TURÁNEK, J. (C2P, s.r.o. – NEXARS, Czech republic): Introduction to theranostics
16:45 - 17:15 CHYTIL, P. (Czech Academy of Science, Czech republic): Synthetic polymers as carriers of biologically active compounds
17:15 - 18:00 BABIČ, M. (Czech Academy of Science, Czech republic): Polymer particles as contrast agents for photoacoustic tomography
18:00 - 18:30 KEŠA, P. (FUJIFILM VisualSonics, Czech republic): High to low-frequency ultrasound and photoacoustic imaging for preclinical research -
19:00 Poster session & Conference banquet
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Friday, September 9, 2022
10:00 - 12:00
Block of Lectures VI
Chairs: prof. CHRISTIAN ZIDORN; assoc. prof. STEFANO DALL'ACQUA
10:00 - 10:45 ZIDORN, CH. (Christian-Albrechts Universität zu Kiel, Germany): Natural products from seagrasses (Alismatales): Chemical diversity, bioactivity, and ecological function
10:45 - 11:30 DALL'ACQUA, S. (University of Padova, Italy): Smart Chain Extraction applied to bark sawmill waste: from research to practical applications
11:30 - 11:45 ŽIGRAYOVÁ, D. (Comenius University Bratislava, Slovakia): Liberation of ibuprofen from polysaccharide hydrogels
11:45 - 12:00 MALANÍK, M. (Masaryk University, Czech republic): A rapid HPLC-ELSD method for separation of sugars and sugar alcohols in fruits of Czech Sorbus species -
12:00 Conference closure